“Transporters, Discovery Metabolism, and Heavy Drugs”

Somerset Crowne Plaza Hotel
110 Davidson Avenue
Somerset, New Jersey

April 22, 2010
8:00 am – 3:30 pm

Program

08:00 am
Registration / Continental Breakfast / Vendor Exhibit

09:00 am
Introductory Remarks
Dr. Philip Krieter, Chair, NJDMDG

09:10 am
Monocarboxylate Transporters in Drug Disposition: Role in the Toxicokinetics and Toxicodynamics of the Drug of Abuse GHB [slides (PDF)] Dr. Marilyn E. Morris, Professor, Department of Pharmaceutical Sciences, University at Buffalo, State University of New York

10:00 am
Disposition and Elimination of Organic Anions and Cations: Transporters and Decision Trees [slides (PDF)] Dr. Douglas H. Sweet, Associate Professor, Department of Pharmaceutics, Virginia Commonwealth University

10:45 am
Vendor Exhibit & Coffee Break

11:15 am
Transporter Polymorphisms [slides (PDF)] Dr. Kathleen Hillgren, Research Advisor, Lilly Research

12:00 pm
Lunch & Vendor Exhibit

01:30 pm
What is Down the Road for Drug Metabolism Support of Drug Metabolism? [slides (PDF)] Dr. Ronald E. White, Distinguished Research Fellow, Pharmaceutical Candidate Optimization, Bristol-Myers Squibb

02:15 pm
Vendor Exhibit & Coffee Break

02:45 pm
Deuterated Drugs: Opportunities and Limitations [slides (PDF)] Dr. Aarti Sawant, Senior Scientist, PDM-CNS Discovery, Pfizer, Inc.

03:45 pm
Program Closure